US 10,010,530 B2
A CARBOXAMIDE DERIVATIVE AND ITS DIASTEREOMERS IN STABLE CRYSTALLINE FORM
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US 10,010,530 B2
A CARBOXAMIDE DERIVATIVE AND ITS DIASTEREOMERS IN STABLE CRYSTALLINE FORM
Tech Center:
1600 Biotechnology and Organic Chemistry
Examiner:
Kamal Saeed
Art Unit:
1626 Organic Chemistry
Agent:
Finnegan, Henderson, Farabow, Garrett & Dunner, L.L.P.
Inventors:
Olli T¿RM¿KANGAS; Terhi HEIKKINEN
Assignee:
ORION CORPORATION
Priority:
01/28/16
Filed:
07/28/17
Granted:
07/03/18
Expiration:
01/28/36
Abstract
The present disclosure relates to solid crystalline forms of N—((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)-propan-2-yl)-5-(1-hydroxyethyl)-1H-pyrazole-3-carboxamide (I) and the diastereomers thereof, and to methods for preparing such crystalline forms. Compound (I) and the diastereomers thereof are potent androgen receptor (AR) modulators useful as a medicament.
Cooperative Patent Classification (CPC)
A61A61P43/00A61K31/4155A61PC07D231/14C07D

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