US 8,329,680 B2
FormulationGeneral
US 8,329,680 B2
Formulation
Tech Center:
1600 Biotechnology and Organic Chemistry
Examiner:
San-Ming Hui
Art Unit:
1629 Organic Chemistry
Inventors:
John R. Evans; Rosalind U. Grundy
Assignee:
Priority:
01/10/00
Filed:
10/15/08
Granted:
12/11/12
Expiration:
01/13/25
Abstract
The invention relates to a novel sustained release pharmaceutical formulation adapted for administration by injection containing the compound 7α-[9-(4,4,5,5,5-pentafluoropentylsulphinyl)nonyl]oestra-1,3,5(10)-triene-3,17β-diol, more particularly to a formulation adapted for administration by injection containing the compound 7α-[9-(4,4,5,5,5-pentafluoropentylsulphinyl)nonyl]oestra-1,3,5(10)-triene-3,17β-diol in solution in a ricinoleate vehicle which additionally comprises at least one alcohol and a non-aqueous ester solvent which is miscible in the ricinoleate vehicle.
Cooperative Patent Classification (CPC)
A61A61K9/0019A61P15/00A61K